{"id":1362,"date":"2026-05-11T22:17:35","date_gmt":"2026-05-12T03:17:35","guid":{"rendered":"https:\/\/elyxaminos.com\/producto\/melanotan-2-10mg\/"},"modified":"2026-07-27T09:33:06","modified_gmt":"2026-07-27T14:33:06","slug":"melanotan-2-10mg","status":"publish","type":"product","link":"https:\/\/elyxaminos.com\/en\/producto\/melanotan-2-10mg\/","title":{"rendered":"Melanotan 2 10mg"},"content":{"rendered":"<section class=\"acordeon\">\n<details open=\"open\">\n<summary>\ud83d\udd39 In-depth Scientific Profile<\/summary>\n<p>Melanotan 2 (MT-2) es un p\u00e9ptido sint\u00e9tico an\u00e1logo de la hormona alfa-melanocito estimulante (\u03b1-MSH), dise\u00f1ado originalmente en la Universidad de Arizona en los a\u00f1os 90 como estrategia para prevenir c\u00e1ncer de piel mediante inducci\u00f3n de bronceado end\u00f3geno previo a exposici\u00f3n solar intensa. Su afinidad por los receptores de melanocortina supera la del \u03b1-MSH natural.<\/p>\n<p><b>Molecular structure:<\/b><\/p>\n<ul>\n<li>Estructura c\u00edclica, lo que extiende su vida media versus \u03b1-MSH lineal<\/li>\n<li>Peso molecular: 1,024 Da<\/li>\n<li>Afinidad alta por MC1R (melanog\u00e9nesis) y MC4R (funci\u00f3n sexual y apetito)<\/li>\n<li>Menor afinidad por MC2R, lo que evita activaci\u00f3n adrenal<\/li>\n<\/ul>\n<\/details>\n<details>\n<summary>\ud83d\udd2c MOLECULAR MECHANISM OF ACTION<\/summary>\n<ul>\n<li><b>Activaci\u00f3n de MC1R en melanocitos:<\/b> estimula la s\u00edntesis de eumelanina, el pigmento responsable del color oscuro y la protecci\u00f3n UV<\/li>\n<li><b>Activaci\u00f3n de MC4R hipotal\u00e1mica:<\/b> reduce apetito y modula funci\u00f3n sexual central<\/li>\n<li><b>Reducci\u00f3n de inflamaci\u00f3n cut\u00e1nea:<\/b> efecto secundario relacionado con su parentesco con \u03b1-MSH<\/li>\n<li><b>Modulaci\u00f3n de termog\u00e9nesis:<\/b> impacto leve sobre gasto energ\u00e9tico basal<\/li>\n<\/ul>\n<\/details>\n<details>\n<summary>\ud83e\uddea RESEARCH APPLICATIONS<\/summary>\n<ul>\n<li>Bronceado seguro previo a exposici\u00f3n solar (research primario original)<\/li>\n<li>Disfunci\u00f3n er\u00e9ctil resistente a inhibidores PDE5<\/li>\n<li>Disfunci\u00f3n del deseo sexual femenino<\/li>\n<li>Vitiligo (investigaciones de repigmentaci\u00f3n)<\/li>\n<li>P\u00e9rdida de peso en investigaciones preliminares<\/li>\n<\/ul>\n<\/details>\n<details>\n<summary>\ud83d\udc89 Reconstitution and Dosage Protocol<\/summary>\n<p><b>Reconstitution<\/b> 2 ml de agua bacteriost\u00e1tica en vial de 10 mg. Concentraci\u00f3n: 5,000 mcg\/ml. Cada unidad U-100 entrega 50 mcg.<\/p>\n<p><b>Fases del protocolo:<\/b><\/p>\n<ul>\n<li><b>Carga (1-3 semanas):<\/b> 250 a 500 mcg\/d\u00eda subcut\u00e1neo (5 a 10 unidades U-100), aumentando gradualmente desde 100 mcg para evaluar tolerancia<\/li>\n<li><b>Mantenimiento:<\/b> 250 a 500 mcg 2 a 3 veces por semana una vez alcanzado el tono deseado<\/li>\n<li><b>Exposici\u00f3n UV controlada:<\/b> 15 a 20 minutos de sol moderado durante fase de carga para potenciar pigmentaci\u00f3n<\/li>\n<\/ul>\n<\/details>\n<details>\n<summary>\u26a0\ufe0f SAFETY CONSIDERATIONS<\/summary>\n<p>Eventos adversos comunes: n\u00e1usea (especialmente primeras dosis), rubor facial, aumento de l\u00edbido, oscurecimiento de lunares preexistentes, aparici\u00f3n de nuevos lunares.<\/p>\n<p><b>Punto cr\u00edtico:<\/b> evaluar dermatol\u00f3gicamente cualquier lunar nuevo o cambio en lunares existentes durante y despu\u00e9s del protocolo. La estimulaci\u00f3n generalizada de melanocitos puede oscurecer lesiones pigmentadas preexistentes, lo que podr\u00eda enmascarar o simular cambios neopl\u00e1sicos.<\/p>\n<p>Contraindicaciones: melanoma activo o sospecha, historia familiar de melanoma sin evaluaci\u00f3n dermatol\u00f3gica previa, embarazo y lactancia.<\/p>\n<\/details>\n<details>\n<summary>\ud83e\uddec STACK Y COMBINACIONES<\/summary>\n<ul>\n<li>MT-2 + PT-141 para frente integral de funci\u00f3n sexual (mecanismos complementarios)<\/li>\n<li>MT-2 + GHK-Cu para soporte cut\u00e1neo durante pigmentaci\u00f3n<\/li>\n<\/ul>\n<\/details>\n<details>\n<summary>\ud83d\udcda SCIENTIFIC REFERENCES<\/summary>\n<ol>\n<li>Dorr RT, Lines R, Levine N, et al. Evaluation of melanotan-II, a superpotent cyclic melanotropic peptide in a pilot phase-I clinical study. Life Sci. 1996;58(20):1777-1784.<\/li>\n<li>Wessells H, Levine N, Hadley ME, Dorr R, Hruby V. Melanocortin receptor agonists, penile erection, and sexual motivation: human studies with Melanotan II. Int J Impot Res. 2000;12 Suppl 4:S74-79.<\/li>\n<li>Hadley ME, Hruby VJ. Discovery and development of novel melanogenic drugs. Pharm Biotechnol. 1998;11:545-575.<\/li>\n<\/ol>\n<\/details>\n<p style=\"margin-top:16px\"><strong>Research material only.<\/strong> This product is intended for scientific research in controlled laboratory settings only. It is not a drug. <strong>Not for human or animal use<\/strong>, not for diagnostic or therapeutic use.<\/p>\n<\/section>","protected":false},"excerpt":{"rendered":"<ul>\n<li>An\u00e1logo sint\u00e9tico de la hormona \u03b1-MSH con afinidad mejorada por receptores MC1R y MC4R.<\/li>\n<li>Investigado en pigmentaci\u00f3n cut\u00e1nea (bronceado) y funci\u00f3n sexual.<\/li>\n<li>Estimulaci\u00f3n de melanog\u00e9nesis natural sin exposici\u00f3n intensa a radiaci\u00f3n UV.<\/li>\n<li>Vial de 10 mg, formato est\u00e1ndar para protocolos de carga y mantenimiento.<\/li>\n<\/ul>\n<p><!-- ELYX-CERT-BUTTONS:start --><\/p>\n<div style=\"display: flex;flex-wrap: wrap;gap: 4px;justify-content: center;margin-top: 24px\">\n<a href=\"https:\/\/elyxaminos.com\/wp-content\/uploads\/2026\/05\/MT2_10MG_COA.pdf\" target=\"_blank\" rel=\"noreferrer\"><button style=\"display: flex;align-items: center;justify-content: center;background: linear-gradient(264.62deg, #02042B 11.77%, #0334D8 62.3%, #48DFE4 91.88%);padding: 15px 30px;border-radius: 50px;color: white;border: none;font-weight: bold;cursor: pointer;text-align: center;font-family: sans-serif;min-width: 150px\">Certificate of Analysis<\/button><\/a><br \/>\n<a href=\"https:\/\/elyxaminos.com\/wp-content\/uploads\/2026\/05\/MT2_10MG_ENDO.pdf\" target=\"_blank\" rel=\"noreferrer\"><button style=\"display: flex;align-items: center;justify-content: center;background: linear-gradient(264.62deg, #02042B 11.77%, #0334D8 62.3%, #48DFE4 91.88%);padding: 15px 30px;border-radius: 50px;color: white;border: none;font-weight: bold;cursor: pointer;text-align: center;font-family: sans-serif;min-width: 150px\">Endotoxins<\/button><\/a>\n<\/div>\n<p><!-- ELYX-CERT-BUTTONS:end --><\/p>","protected":false},"featured_media":1578,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[35],"product_tag":[],"class_list":{"0":"post-1362","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-sexual-health","8":"first","9":"instock","10":"shipping-taxable","11":"purchasable","12":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/product\/1362","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/comments?post=1362"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/media\/1578"}],"wp:attachment":[{"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/media?parent=1362"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/product_brand?post=1362"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/product_cat?post=1362"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/elyxaminos.com\/en\/wp-json\/wp\/v2\/product_tag?post=1362"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}